Publications 2001-2010

2010 / 2009 / 2008 / 2007 / 2006 / 2005 / 2004 / 2003 / 2002 / 2001

2010

Structure Elucidation of Dimethylformamide-Solvated Alkylzinc Cations in the Gas Phase.

Dreiocker, Frank; Oomens, Jos; Meijer, Anthony J. H. M.; Pickup, Barry T.; Jackson, Richard F. W.; Schafer, Mathias.

J. Org. Chem.201075, 1203-1213.

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Much Improved Conditions for the Negishi Cross-Coupling of Iodoalanine Derived Zinc Reagents with Aryl Halides

Ross, Andrew J.; Lang, Hannah L.; Jackson, Richard F. W.

J. Org. Chem., 2010, 75, 245-248.

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Improved synthesis of phenylethylamine derivatives by Negishi cross-coupling reactions

Goddard, Craig M. L.; Massah, Ahmad Reza; Jackson, Richard F. W.

Tetrahedron, 2010, 66, 9175-9181.

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In situ trapping of Boc-2-pyrrolidinylmethylzinc iodide with aryl iodides: direct synthesis of 2-benzylpyrrolidines

Massah, Ahmad Reza; Ross, Andrew J.; Jackson, Richard F. W.

J. Org. Chem., 2010, 75, 8275-8278.

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2009

An approach to the synthesis of anti-β-2,3-amino acids: application of β-trifluoroacetamidoorganozinc reagents.

Bartrum, Hannah E.; Jackson, Richard F. W.

Synlett, 2009, 2257

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Enantioselective Oxidation of an Alkyl Aryl Sulfide: Synthesis of (S)-(-)-Methyl p-Bromophenyl Sulfoxide.

Drago, Carmelo; Walker, Emma-Jane; Caggiano, Lorenzo; Jackson, Richard F. W.

Organic Syntheses, 2009, 86, 121-129.

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Recent Developments in the Application of Organometallic Chemistry to Amino Acid Synthesis

Jackson, R. F. W.

In Asymmetric Synthesis and Application of α-Amino Acids; Soloshonok, V. A., Izawa, K., Eds.; American Chemical Society: Washington, DC, 2009, p 2-12.


Application of Negishi Cross-Coupling to the Synthesis of the Cyclic Tripeptides OF4949-III and K-13.

Nolasco, Luca; Perez Gonzalez, Manuel; Caggiano, Lorenzo; Jackson, Richard F. W.

J. Org. Chem., 2009, 74, 8280-8289

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Crystal structure of 2-(4-methoxybenzylthio)-1-phenylethanone.

Heravi, Mohammad R. Poor; Loghmani-Khouzani, Hossein; Sadeghi, Majid M. M.; Zendehdel, Mahmoud; Jackson, Richard F. W.

Analytical Sciences: X-Ray Structure Analysis Online, 2009, 25, 43

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2008

Negishi cross-coupling reactions of α-amino acid-derived organozinc reagents and aryl bromides

Oswald, Claire L.; Carrillo-Márquez, Tomás; Caggiano, Lorenzo; Jackson, Richard F. W.

Tetrahedron, 2008, 64, 681-687.

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Investigation of a Flexible Enantiospecific Approach to Aziridines

Jamookeeah, Clare E.; Beadle, Christopher D.; Jackson, Richard F. W.; Harrity, Joseph P. A.

J. Org. Chem., 2008, 73, 1128-1130.

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Synthesis of β2-homophenylalanine derivatives by Negishi cross-coupling reactions

Bartrum, Hannah E.; Adams, Harry; Caggiano, Lorenzo; Jackson, Richard F. W.

Tetrahedron, 2008, 64, 3701-3712.

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α-Fluorination of β-ketosulfones by Selectfluor™(F-TEDA-BF4)

Loghmani-Khouzani, Hossein; Poorheravi, Mohammad R.; Sadeghi, Majid M. M.; Caggiano, Lorenzo; Jackson, Richard F. W.

Tetrahedron, 2008, 64, 7419–7425.

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Ionisation of the Zinc-Iodine Bond of Alkylzinc Iodides in Dimethylformamide from Theory and Experiment

Caggiano, Lorenzo; Jackson, Richard F. W.; Meijer, Anthony J. H. M.; Pickup, Barry T.; Wilkinson, Karl A.

Chem. Eur. J., 2008, 14, 8798-8802.

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Kinetic Studies on the Stability and Reactivity of β-Amino Alkylzinc Iodides Derived from Amino Acids

Rilatt, Ian; Jackson, Richard F. W.

J. Org. Chem., 2008, 73, 8694-8704.

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2007

Stereoselective synthesis of 2,3-difunctionalised thioesters using nucleophilic epoxidation of 1-arylthio-1-nitroalkenes

Evans, Lyndsay Ann; Adams, Harry; Barber, Christopher G.; Caggiano, Lorenzo; Jackson, Richard F. W.

Org. Biomol. Chem., 2007, 5, 3156-3163.

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2006

Effective Asymmetric Oxidation of Enones and Alkyl Aryl Sulfides

Hinch, Melissa; Jacques, Olivier; Drago, Carmelo; Caggiano, Lorenzo; Jackson, Richard F. W.

J. Mol. Cat. A: Chemical, 2006, 251, 123-128.

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Synthesis of Orthogonally Protected Biaryl Amino Acid Derivatives

Moreno, Eduardo; Nolasco, Luca Antonio; Caggiano, Lorenzo; Jackson, Richard F. W.

Org. Biomol. Chem., 2006, 4, 3639-3647.

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Oxidative Kinetic Resolution of Alkyl Aryl Sulfoxides

Mohammadpoor-Baltork, Iraj; Hill, Mathias; Caggiano, Lorenzo; Jackson, Richard F. W.

Synlett, 2006, 3540-3544.

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2005

New Routes to β-Cycloalkylalanine Derivatives using Serine-Derived Organozinc Reagents

Carrillo-Marquez, Tomas; Caggiano, Lorenzo; Jackson, Richard F. W.; Grabowska, Urszula; Rae, Alastair; Tozer, Matthew J.

Org. Biomol. Chem., 2005, 3, 4117 - 4123.

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Development and Applications of Amino Acid-Derived Organometallics

Rilatt, Ian; Caggiano, Lorenzo; Jackson, Richard F. W.

Synlett, 2005, 2701-2719.

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Vanadium-Catalysed Sulfur Oxidation/Kinetic Resolution Process for the Synthesis of Enantiomerically Pure Alkyl Aryl Sulfoxides

Drago, Carmelo; Caggiano, Lorenzo; Jackson, Richard F. W.

Angew. Chem. Int Ed. Engl., 2005, 7221-7223.

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2004

Synthesis of Unprotected Phenols using Palladium-Catalysed Cross Coupling Reactions of Functionalised Organozinc Reagents

Jackson, Richard F. W.; Rilatt, Ian; Murray, P. John

Org. Biomol. Chem., 2004, 2, 110-113.

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Synthesis of N-(tert-Butoxycarbonyl)-β-Iodoalanine Methyl Ester: A Useful Building Block in the Synthesis of Nonnatural α-Amino Acids via Palladium Catalysed Cross Coupling Reactions

Jackson, Richard F. W.; Perez-Gonzalez, Manuel

Org. Synth., 2004, 81, 77-87.

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2003

Benzyl (2S)-2-tert-butoxycarbonylamino-5-(2-furyl)-5- oxopentanoate

Clegg, William, Wishart, Neil; Jackson, Richard F. W.

Acta Crystallogr. Sect. E.-Struct Rep. Online, 2003, O86-O88.

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Cross coupling reactions of organozinc iodides with solid- supported electrophiles: synthesis of 4-substituted benzoic and 3-substituted (E)- and (Z)-propenoic acids and amides

Oates, Leslie J.; Jackson, Richard F. W.; Block, Michael H.

Org. Biomol. Chem. , 2003, 1, 140-144.

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Combined application of organozinc chemistry and one-pot hydroboration-Suzuki coupling to the synthesis of amino acids

Rodriguez, Arantxa; Miller, David D.; Jackson, Richard F. W.

Org. Biomol. Chem., 2003, 1, 973-977.

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The rate of elimination of a β-amino zinc reagent is reduced by using a better leaving group

Jackson, Richard F. W.; Rilatt, Ian; Murray, P. John

Chem. Commun., 2003, 1242-1243.

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Synthesis and crystal structures of 2-substituted-2-phenylsulfonyloxiranes: evidence for a generalised anomeric effect in 2-phenylsulfonyloxiranes

Jackson, Richard F. W.; Dunn, Sara F. C.; McCamley, Andrew; Clegg, William

Org. Biomol. Chem., 2003, 1, 2527-2530.

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[3 R-(3b,4b,5b)]-3-(Acetylamino)-3,4-dihydro-4-hydroxy-5-(hydroxymethyl) furan-2(5H)-one monohydrate

Clegg, William; Heath, Sarah L.; Jackson, Richard F. W.; Palmer, Nicholas J.

Acta Crystallogr. Sect. E.-Struct Rep. Online, 2003, 59, O1060-O1062.

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Preparation of Enantiomerically Pure Pyridyl Amino Acids from Serine

Tabanella, Stefania; Valancogne, Ingrid; Jackson, Richard F. W.

Org. Biomol. Chem., 2003, 1, 4254-4261.

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2002

Synthesis of 2-Substituted Indolines using Sequential Pd-Catalyzed Processes

Deboves, Hervé J. C.; Hunter, Christopher; Jackson, Richard F. W.

J. Chem. Soc., Perkin Trans 1, 2002, 733-736.

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Synthesis of Macrocyclic, Potential Protease Inhibitors using a Generic Scaffold

Dumez, Estelle; Snaith, John S.; Jackson, Richard F. W.; McElroy, Andrew B.; Overington, John; Wythes, Martin J.; Withka, Jane M.; McLellan, Thomas J.

J. Org. Chem., 2002, 67, 4882-4892.

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Enantioselective Sulfide Oxidation with H2O2; A Solid Phase and Array Approach for the Optimisation of Chiral Schiff Base-Vanadium Catalysts

Pelotier, Béatrice; Anson, Mike S.; Campbell, Ian B.; Macdonald, Simon J.F.; Priem, Ghislaine; Jackson, Richard F.W.

Synlett, 2002, 1055-1060.

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Asymmetric Michael Reactions Using Tartrate-based Magnesium Catalysts

MacCulloch, Alasdair C.; Yolka, Sylvie; Jackson, Richard F.W.

Synlett, 2002, 1700-1702.

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Stereocontrolled Synthesis of anti-α-Hydroxy-β-Amino and anti-α,β-Diamino Acid Derivatives by Epoxidation of 1-Arylthio-1-nitroalkenes

Ambroise, Lydia; Dumez, Estelle; Szeki, Andrea; Jackson, Richard F. W.

Synthesis, 2002, 2296-2308.

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Palladium(0) catalysed and copper(I) promoted reactions of the secondary zinc reagent derived from L-threonine

Wilson, Ian; Jackson, Richard F. W.

J. Chem. Soc., Perkin Trans 1, 2002, 2845-2850.

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2001

Synthesis of a 3-aminopiperidin-2,5-dione as a conformationally constrained surrogate of the Ala-Gly dipeptide

Estiarte, M. Angels; Diez, Anna; Rubiralta, Mario; Jackson, Richard F.W.

Tetrahedron, 2001, 57, 157-161.

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Optimization of new chiral ligands for the copper-catalysed enantioselective conjugate addition of Et2Zn to nitroolefins by high-throughput screening of a parallel library

Ongeri, Sandrine; Piarulli, Umberto; Jackson, Richard F. W.; Gennari, Cesare

Eur. J. Org. Chem., 2001, 803-807.

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Improved catalytic procedures for the copper(I)-promoted reactions of β-amido zinc reagents

Hunter, Christopher; Jackson, Richard F. W.; Rami, Harshad K.

J. Chem. Soc., Perkin Trans 1, 2001, 1349-1352.

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Direct Synthesis of Fmoc-protected Amino Acids using Organozinc Chemistry: Application to Polymethoxylated Phenylalanines and 4-Oxo Amino Acids

Deboves, Hervé J. C.; Montalbetti, Christian A. G. N.; Jackson, Richard F. W.

J. Chem. Soc., Perkin Trans 1, 2001, 1876-1884.

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Stereoselective Synthesis of Differentially Protected anti-α,β-Diamino Acid Derivatives using Arylthionitrooxiranes

Dumez, Estelle; Szeki, Andrea; Jackson, Richard F. W.

Synlett, 2001, 1214-1216.

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Discovery of New Solid Phase Sulfur Oxidation Catalysts using Library Screening

Green, Stuart D.; Monti, Chiara; Jackson, Richard F. W.; Anson, Michael S.; Macdonald, Simon J. F.

Chem. Commun., 2001, 2954-2955.

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Catalytic Asymmetric Epoxidation of Aliphatic Enones using Tartrate-derived Magnesium Alkoxides

Jacques, Olivier; Richards, Sarah J.; Jackson, Richard F. W.

Chem. Commun., 2001, 2712-2713.

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